Addition of indoles to oxyallyl cations for facile access to α-indole carbonyl compounds.
نویسندگان
چکیده
A direct coupling of unprotected indoles and α-halo ketones via in situ generated oxyallyl cation intermediates is described. The reactions efficiently afford α-indole carbonyl compounds with good to quantitative yields.
منابع مشابه
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ورودعنوان ژورنال:
- Organic letters
دوره 14 7 شماره
صفحات -
تاریخ انتشار 2012